LA Pharma Cypionate 1 ml vial (200 mg/ml) EXPIRATION

Testosterone Cypionate

Is a long-acting testosterone formulation indicated for individuals with low or absent hormone levels, often referred to as Depo-Testosterone. This esterified form of testosterone is exclusively available for injection and is usually dissolved in sesame or cottonseed oil. Gradually released from the injection site, its effects can last between 7 to 12 days. The formulation appears as a white milky powder, insoluble in water but easily dissolvable in most organic solvents, including vegetable oil.

Pharmacology

The body naturally produces hormones like testosterone, crucial for the growth and development of secondary sexual characteristics such as the prostate, testes, penis, scrotum, body hair, and muscle mass. Testosterone therapy is often necessary for individuals experiencing testosterone deficiency, which can lead to abnormal development of these characteristics.

Indications for Use

Testosterone Cypionate treats conditions related to inadequate secretion of testosterone, including:

• Primary testicular failure
• Failure of the pituitary gland to release gonadotropins

Bodybuilding

Both athletes and bodybuilders commonly utilize testosterone and its derivatives to enhance performance and boost motivation. Many users report bursts of energy and heightened aggression, especially in activities like weightlifting and professional wrestling. While testosterone has moderate anabolic effects, it is also a powerful androgen. As an injectable solution, its benefits are not immediate, with effects typically seen after 3-4 weeks, lasting longer than oral formulations. A diet rich in calories is essential for muscle building while using testosterone. Bodybuilders often stack it with other hormones, and due to its conversion to estrogen, there’s a risk of gynecomastia and water retention. To mitigate these effects, compounds like Arimidex or tamoxifen are usually employed during off-cycles.

Contraindications

Certain individuals should avoid testosterone due to potential aggravation of specific conditions, including:

• Allergic reactions to the drug
• Males with breast or prostate cancer
• Pregnant or breastfeeding women
• Individuals with heart, liver, or kidney diseases

Side Effects

When injected in low doses, side effects of Testosterone Cypionate are rare. Long-term usage can be associated with various reversible side effects, although for females, virilizing effects may be permanent. Common side effects include:

• Nausea and vomiting
• Abdominal cramps and diarrhea
• Swelling
• Changes in libido
• Headaches
• Acne and oily skin
• Mood changes including aggression, depression, and insomnia
• Excessive sweating
• Hair loss
• Gynecomastia

For females, virilizing effects may manifest as:

• Voice deepening
• Hoarseness
• Excessive body hair growth
• Enlarged clitoris
• Irregular menstrual cycles

Hormonal conversion in fat tissue can lead to estrogen-related developments like breast enlargement and fluid retention, especially after prolonged use of over 4 weeks, with gynecomastia being reversible upon discontinuation.

Overdose

Overdosing on Testosterone Cypionate is infrequent. While overdose from injection typically does not produce acute symptoms, individuals may experience illness lasting weeks. Medical consultation may be advisable for excessive doses.

Dosage

In clinical practice, Testosterone Cypionate is administered via intramuscular injection, available in strengths of 100 mg/ml and 200 mg/ml. Injections occur in the buttock every 7 to 12 days. Although the drug normally binds to proteins with only 2% remaining free, some bodybuilders opt for more frequent dosing every other day, which could lead to complications such as abscesses or infections if not administered correctly. Injection sites should be alternated for prolonged use, with dosages typically ranging from 50 mg to 400 mg per week, higher for bodybuilding purposes (200 mg to 400 mg weekly). The release into the bloodstream is gradual over days.

Control

Testosterone Cypionate is classified as a controlled substance (Class 3) under the Controlled Substance Act in the USA, requiring a physician’s prescription for legal acquisition. Possession or distribution without a prescription is illegal.

Detection

The oily suspension of Testosterone Cypionate can remain detectable in urine for 2-3 weeks post-injection, which leads many bodybuilders to use it primarily during off-seasons.

Availability

Many bodybuilders source Testosterone Cypionate from the black market, as pharmaceutical options in the USA are highly regulated. Generic versions are produced in various countries, including Japan, Australia, Mexico, Spain, Brazil, and Thailand, with usage rates ranging from 200-1000 mg/week. Prices can vary, with a 400 mg vial costing between $20-$40, potentially totaling up to $200 monthly. However, product purity and authenticity can be questionable, with counterfeit products widely available.