PharmARC Cypiosteron 6 amps (6x 250 mg/ml)

Testosterone Cypionate

Is a long-acting testosterone formulation indicated for individuals with critically low or absent levels of this essential hormone, also known as Depo Testosterone. This esterified form provides extended effects through intramuscular injection, typically utilizing sesame or cottonseed oil as a solvent, allowing for a sustained release of testosterone lasting from 7 to 12 days.

The drug appears as a white, milky powder, insoluble in water but readily dissolvable in most organic solutions, including vegetable oils.

Pharmacology

The body naturally produces sex hormones like testosterone, crucial for developing secondary sexual characteristics such as prostate and testes growth, body hair, and specific fat distribution. Testosterone deficiency can lead to abnormal bodily growth and secondary characteristics. Hence, testosterone therapy is vital for individuals with low testosterone levels and those facing infertility challenges.

Indications for Use

Testosterone Cypionate is utilized for conditions resulting from inadequate testosterone secretion, including:

• Primary testicular failure
• Pituitary insufficiency in releasing Gonadotropins

Bodybuilding

Testosterone and its derivatives are popular among athletes and bodybuilders for their ability to enhance physical performance and energy levels. Users often report increased aggression and energy bursts, particularly beneficial for weightlifters and wrestlers. Despite moderate anabolic properties, testosterone is recognized as a potent androgenic agent.
The onset of effects is gradual post-injection, typically taking 3-4 weeks, although injected formulations can last longer in the system compared to oral alternatives. Long-term usage over 4-6 weeks can boost body mass and protein synthesis, provided the individual maintains a calorie-rich diet. Bodybuilders often combine testosterone with other hormones, but care is needed to manage potential estrogen conversion, which can lead to gynecomastia and water retention. To mitigate these effects, agents like Arimidex or tamoxifen are commonly included in cycling plans.
Regular injections can inhibit natural testosterone production through the feedback mechanism, potentially impacting spermatogenesis at higher doses. Gradual tapering over several weeks is recommended to allow recovery of the hypothalamic-pituitary axis, as abrupt cessation may lead to fatigue, weight loss, and increased fracture risk.

Contraindications

Certain individuals should avoid testosterone due to potential exacerbation of medical conditions, including:

• Allergic reactions to the substance
• Males with breast or prostate cancer
• Women who are pregnant or nursing
• Individuals with liver, kidney, or heart disease

Side Effects

At lower doses, Testosterone Cypionate generally has minimal side effects, but prolonged use may cause reversible adverse effects. Women taking testosterone might face irreversible virilizing effects. Common side effects include:

• Nausea, vomiting
• Abdominal discomfort
• Fluid retention
• Altered libido
• Headaches
• Acne and oily skin
• Mood changes such as aggression and depression
• Increased sweating
• Hair loss
• Gynecomastia

For women, additional virilizing effects may consist of:

• Deepening voice
• Hoarseness
• Excessive hair growth
• Enlargement of clitoris
• Irregular menstrual cycles

Conversion to estrogen can cause breast enlargement and water retention, potentially noticeable after 4 weeks of use, though these effects usually reverse upon discontinuation.

Overdose

Instances of overdose with Testosterone Cypionate are rare, typically presenting as mild illness without acute side effects. Medical consultation is advisable following any suspected overdose.

Dosage

In clinical settings, Testosterone Cypionate is administered via intramuscular injection in oily suspension form, available in 100mg/ml and 200mg/ml strengths. Recommended injection sites are the buttocks every 7-12 days, although some bodybuilders may choose more frequent doses, which can lead to complications like abscesses if not managed properly. Typical dosages range from 50mg to 400mg per week, with bodybuilders usually opting for higher doses between 200mg and 400mg weekly.

Control

Regulated under Class 3 of the Controlled Substances Act, Testosterone Cypionate requires a valid physician’s prescription for legal possession and distribution in the USA.

Detection

As an oily drug suspension, its metabolites can linger in the body, detectable for up to 2-3 weeks post-injection. This prolonged presence often leads bodybuilders to use it seasonally.

Availability

Many bodybuilders source Testosterone Cypionate via the black market, as legitimate pharmaceutical products are highly regulated in the USA. Generic variants are produced in countries like Japan, Australia, and Mexico. Prices may range from $20-$40 for 400mg vials, potentially summing to $200 monthly, depending on usage. It’s essential to be cautious of product purity and potential forgery in such markets.